Nattokinase

Bacillus subtilis natto
Evidence Level
Moderate
2 Clinical Trials
5 Documented Benefits
3/5 Evidence Score

Nattokinase is a fibrinolytic enzyme produced by Bacillus subtilis natto fermentation of soybeans (the traditional Japanese food natto). Distinguished by ability to break down fibrin (blood clots) — the only oral enzyme with substantial human data on cardiovascular and circulation effects. Used for cardiovascular support, deep vein thrombosis prevention, and recently long-COVID/post-vaccination spike protein concerns. Standardized in fibrinolytic units (FU).

Studied Dose 100-400 mg/day standardized to 2,000-8,000 FU (fibrinolytic units); typically taken on empty stomach
Active Compound Nattokinase (subtilisin NK, serine protease)

Benefits

Fibrinolytic Activity

Nattokinase directly cleaves fibrin (the protein scaffold of blood clots) — distinct from anticoagulants (which prevent clot formation by inhibiting clotting factors) and antiplatelets (which prevent platelet aggregation). Activates endogenous tissue plasminogen activator (tPA) and degrades fibrin directly.

Blood Pressure Modest Reduction

Kim 2008 and Jensen 2016 RCTs showed nattokinase (2,000 FU/day) modestly reduced both systolic and diastolic blood pressure in pre/hypertensive adults vs placebo. Effect size ~5-6 mmHg systolic — clinically meaningful but modest.

Cardiovascular Risk Markers

Several trials show nattokinase reduces fibrinogen, factor VII, and factor VIII levels — plus may reduce LDL and triglycerides, raise HDL. Multi-mechanism cardiovascular support.

Deep Vein Thrombosis (DVT) Prevention (Theoretical)

Cesarone 2003 trial showed nattokinase (2 capsules/day) reduced edema and DVT incidence vs placebo on long-haul flights. Mechanism plausible; sample size limited. Standard DVT prevention for high-risk patients remains anticoagulants and compression.

Long-COVID / Spike Protein Research (Emerging)

Recent in vitro research (Tanikawa 2022) suggests nattokinase may degrade SARS-CoV-2 spike protein. Generated significant interest in long-COVID and post-vaccine spike protein clearance. CRITICAL CAVEAT: in vitro evidence; human clinical translation not established; do NOT use as substitute for evidence-based COVID treatments.

Mechanism of action

1

Direct Fibrin Cleavage

Nattokinase is a serine protease that directly cleaves fibrin into smaller fragments — same end result as endogenous plasmin. Distinct from anticoagulant drugs (which work upstream by inhibiting clotting factors).

2

tPA Activation

Nattokinase enhances production and activity of endogenous tissue plasminogen activator (tPA) — increasing physiological fibrinolytic capacity. Both direct (NK cleaves fibrin) and indirect (NK activates plasmin via tPA) mechanisms.

3

PAI-1 Inhibition

Nattokinase reduces plasminogen activator inhibitor-1 (PAI-1) — a fibrinolysis inhibitor. Lower PAI-1 = greater fibrinolytic activity. PAI-1 elevation associated with metabolic syndrome and CV risk.

4

Pleiotropic Cardiovascular Effects

Beyond fibrinolysis: BP reduction (mechanism unclear; possibly via ACE inhibition), modest lipid effects, reduced platelet aggregation. Multi-mechanism CV agent.

Clinical trials

1
Nattokinase for Hypertension — Kim 2008
PubMed

Double-blind RCT of nattokinase (2,000 FU/day) vs placebo in 86 prehypertensive adults for 8 weeks.

86 prehypertensive adults.

Nattokinase reduced systolic BP by ~5.5 mmHg and diastolic BP by ~2.8 mmHg vs placebo. Modest but clinically meaningful effect. Subsequent Jensen 2016 trial confirmed similar magnitude.

2
Nattokinase for DVT Prevention (Long-Flight) — Cesarone 2003
PubMed

RCT of nattokinase + pycnogenol vs placebo for DVT prevention in 200 long-haul flight passengers.

200 high-risk flight passengers.

Nattokinase + pycnogenol group: 0% DVT incidence vs 5% in placebo group; significant edema reduction. Combined product limits attribution to nattokinase alone. Suggestive but not definitive.

About this ingredient

About the active ingredient

Nattokinase is a SERINE PROTEASE (subtilisin NK) produced by Bacillus subtilis natto fermentation of soybeans — the enzyme responsible for the slimy, stringy texture of traditional Japanese natto food. Distinguished from other proteolytic enzymes by SPECIFIC FIBRIN-DEGRADING activity. Standardized in FIBRINOLYTIC UNITS (FU) — typical clinical dose: 2,000-8,000 FU/day (~100-400 mg standardized extract). DISTINCT FROM ANTICOAGULANTS: anticoagulants (warfarin, DOACs) prevent clot FORMATION by inhibiting clotting factors; nattokinase BREAKS DOWN existing fibrin — different mechanism, different clinical use.

EVIDENCE-BASED USES: (1) Modest BP reduction (Kim 2008, Jensen 2016 — ~5 mmHg systolic); (2) Cardiovascular risk marker improvement (fibrinogen, factor VII/VIII, lipids); (3) DVT prevention adjunct (Cesarone 2003 — small trial, combined product); (4) Post-thrombotic syndrome adjunct (limited evidence); (5) Cardiovascular general support. EMERGING/CONTROVERSIAL: (6) LONG-COVID and post-vaccine spike protein concerns — Tanikawa 2022 IN VITRO evidence only; no human clinical trials; do NOT substitute for evidence-based COVID care.

CRITICAL CAUTIONS: (1) BLEEDING RISK — fibrinolytic activity carries bleeding risk; (2) ANTICOAGULANT/ANTIPLATELET COMBINATION — additive bleeding risk; warfarin INR monitoring essential; consult prescriber before combining; (3) PRE-SURGERY — discontinue 1-2 weeks before any surgery; (4) ACTIVE BLEEDING, GI ULCERS, INTRACRANIAL HEMORRHAGE history — AVOID; (5) PREGNANCY/LACTATION — insufficient safety data; AVOID; (6) RECENT STROKE — type-dependent; consult neurologist; (7) SOYBEAN ALLERGY — theoretical cross-reactivity (residual soy protein in standardized products typically very low); (8) ENTERIC COATING — improves stability through gastric acid; some products use enteric coating; (9) STORAGE — heat and acid stability issues; product quality varies; choose reputable brands with FU standardization; (10) DOSE — 2,000 FU is most-studied clinical dose; higher doses (4,000-8,000 FU) used for cardiovascular indications; (11) The 'natural blood thinner' marketing is somewhat misleading — nattokinase is fibrinolytic (clot-busting) rather than anticoagulant; (12) For ESTABLISHED CVD, evidence-based pharmacotherapy (ACEi/ARB, beta-blockers, antiplatelets, statins) remains foundational; nattokinase adjunctive at most.

Side effects and drug interactions

Common Potential side effects

BLEEDING RISK — fibrinolytic activity carries theoretical bleeding risk; particular concern with anticoagulants/antiplatelets, recent surgery, GI ulcers, intracranial bleeding history.
GI distress at high doses.
Headache.
Allergic reactions (rare; soybean source).
Skin reactions rare.
PRE-SURGERY DISCONTINUATION — discontinue 1-2 weeks before any surgery to reduce bleeding risk.

Important Drug interactions

ANTICOAGULANTS (warfarin, apixaban, rivaroxaban, dabigatran, edoxaban, heparin) — additive bleeding risk; CONSULT prescriber; INR monitoring with warfarin essential; avoid concurrent without medical supervision.
ANTIPLATELET drugs (aspirin, clopidogrel, prasugrel, ticagrelor) — additive bleeding risk; consult cardiologist.
Fibrinolytic drugs (tPA, alteplase, streptokinase) — additive; not relevant for chronic outpatient use.
NSAIDs — additive bleeding risk especially with chronic use.
Fish oil, garlic, ginkgo, vitamin E (high-dose) — multiple supplements have antiplatelet effects; cumulative bleeding risk.
Soybean allergy — nattokinase is derived from fermented soy; theoretical cross-reactivity (typically very low residual soy protein in standardized products).

Frequently asked questions about Nattokinase

What is the recommended dosage of Nattokinase?

The clinically studied dose for Nattokinase is 100-400 mg/day standardized to 2,000-8,000 FU (fibrinolytic units); typically taken on empty stomach. Always follow product labeling and consult a healthcare provider for personalized dosing recommendations.

What is Nattokinase used for?

Nattokinase is studied for fibrinolytic activity, blood pressure modest reduction, cardiovascular risk markers. Nattokinase directly cleaves fibrin (the protein scaffold of blood clots) — distinct from anticoagulants (which prevent clot formation by inhibiting clotting factors) and antiplatelets (which prevent platelet aggregation).

Are there side effects from taking Nattokinase?

Reported potential side effects may include: BLEEDING RISK — fibrinolytic activity carries theoretical bleeding risk; particular concern with anticoagulants/antiplatelets, recent surgery, GI ulcers, intracranial bleeding history. GI distress at high doses. Always consult a healthcare provider before starting any new supplement, especially if you have underlying conditions or take medications.

Does Nattokinase interact with medications?

Known drug interactions may include: ANTICOAGULANTS (warfarin, apixaban, rivaroxaban, dabigatran, edoxaban, heparin) — additive bleeding risk; CONSULT prescriber; INR monitoring with warfarin essential; avoid concurrent without medical supervision. ANTIPLATELET drugs (aspirin, clopidogrel, prasugrel, ticagrelor) — additive bleeding risk; consult cardiologist. Consult a pharmacist or healthcare provider if you take prescription medications.

Is Nattokinase good for cardiovascular?

Yes, Nattokinase is researched for Cardiovascular support. Kim 2008 and Jensen 2016 RCTs showed nattokinase (2,000 FU/day) modestly reduced both systolic and diastolic blood pressure in pre/hypertensive adults vs placebo. Effect size ~5-6 mmHg systolic — clinically meaningful but modest.